Search on: AGENTS, CALCIMIMETIC 
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Descriptor English:   Calcimimetic Agents 
Descriptor Spanish:   Calcimiméticos 
Descriptor Portuguese:   Calcimiméticos 
Synonyms English:   Agents, Calcimimetic  
Tree Number:   D06.347.230
D27.505.696.399.450.230
Definition English:   Small organic molecules that act as allosteric activators of the calcium sensing receptor (CaSR) in the PARATHYROID GLANDS and other tissues. They lower the threshold for CaSR activation by extracellular calcium ions and diminish PARATHYROID HORMONE (PTH) release from parathyroid cells. 
History Note English:   2011 
Allowable Qualifiers English:  
AD administration & dosage AE adverse effects
AG agonists AN analysis
BL blood CF cerebrospinal fluid
CS chemical synthesis CH chemistry
CL classification CT contraindications
EC economics HI history
IM immunology IP isolation & purification
ME metabolism PK pharmacokinetics
PD pharmacology PO poisoning
RE radiation effects ST standards
SD supply & distribution TU therapeutic use
TO toxicity UR urine
Record Number:   54038 
Unique Identifier:   D057966 

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